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Prof. Dr.  Philipp Heretsch

https://orcid.org/0000-0002-9967-3541
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Publications

  1. 2023

  2. Published

    Biogenetic space-guided synthesis of rearranged terpenoids

    Alekseychuk, M. & Heretsch, P., 10 May 2023, In: Chemical communications. 59, 45, p. 6811-6826 16 p.

    Research output: Contribution to journal › Article › Research › peer review

  3. Published

    Biogenesis-Inspired Synthesis of Penicillitone

    Heretsch, P. & Bauer, M., 23 Feb 2023, In: Synthesis. 55, 9, p. 1322-1327 6 p.

    Research output: Contribution to journal › Article › Research › peer review

  4. Published

    Modern flow chemistry – prospect and advantage

    Heretsch, P., 6 Jan 2023, In: Beilstein Journal of Organic Chemistry. 19, p. 33-35 3 p.

    Research output: Contribution to journal › Editorial in journal › Research › peer review

  5. 2022

  6. Published

    Chemical Emulation of the Biosynthetic Route to Anthrasteroids: Synthesis of Asperfloketal A

    Alekseychuk, M. & Heretsch, P., 7 Dec 2022, In: Journal of the American Chemical Society. 144, 48, p. 21867-21871 5 p.

    Research output: Contribution to journal › Article › Research › peer review

  7. Published

    Biogenesis-Inspired, Divergent Synthesis of Spirochensilide A, Spirochensilide B, and Abifarine B Employing a Radical-Polar Crossover Rearrangement Strategy

    Alekseychuk, M., Adrian, S., Heinze, R. C. & Heretsch, P., 6 Jul 2022, In: Journal of the American Chemical Society. 144, 26, p. 11574-11579 6 p.

    Research output: Contribution to journal › Article › Research › peer review

  8. Published

    Synthesis of odorants in flow and their applications in perfumery

    Kleoff, M., Kiler, P. & Heretsch, P., 2022, In: Beilstein Journal of Organic Chemistry. 18, p. 754-768 15 p.

    Research output: Contribution to journal › Review article › Research › peer review

  9. 2021

  10. External

    A Modular, Argon-Driven Flow Platform for Natural Product Synthesis and Late-Stage Transformations

    Kleoff, M., Schwan, J., Christmann, M. & Heretsch, P., 19 Mar 2021, In: Organic letters. 23, 6, p. 2370-2374 5 p.

    Research output: Contribution to journal › Article › Research › peer review

  11. External

    Scalable Synthesis of Benzotriazoles via [3+2] Cycloaddition of Azides and Arynes in Flow

    Kleoff, M., Boeser, L., Baranyi, L. & Heretsch, P., 8 Feb 2021, In: European Journal of Organic Chemistry. 2021, 6, p. 979-982 4 p.

    Research output: Contribution to journal › Article › Research › peer review

  12. 2020

  13. External

    Synthetic strategies for the ibophyllidine alkaloids

    Reuss, F. & Heretsch, P., 19 Oct 2020, In: Natural product reports. 38, 4, p. 693-701 9 p.

    Research output: Contribution to journal › Article › Research › peer review

  14. External

    Discoveries and Challenges en Route to Swinhoeisterol A

    Duecker, F. L., Heinze, R. C., Steinhauer, S. & Heretsch, P., 7 Aug 2020, In: Chemistry - A European Journal. 26, 44, p. 9971-9981 11 p.

    Research output: Contribution to journal › Article › Research › peer review

  15. External

    Taxane Meets Propellane: First Chemical Synthesis of Highly Complex Diterpene Canataxpropellane

    Reuss, F. & Heretsch, P., 15 Jun 2020, In: Angewandte Chemie - International Edition. 59, 26, p. 10232-10234 3 p.

    Research output: Contribution to journal › Editorial in journal › Research › peer review

  16. External

    Synthesis of Aspidodispermine via Pericyclic Framework Reconstruction

    Reuss, F. & Heretsch, P., 15 May 2020, In: Organic letters. 22, 10, p. 3956-3959 4 p.

    Research output: Contribution to journal › Article › Research › peer review

  17. External

    Synthesis of the Alleged Structures of Fortisterol and Herbarulide and Structural Revision of Herbarulide

    Duecker, F. L., Heinze, R. C., Mueller, M., Zhang, S. & Heretsch, P., 21 Feb 2020, In: Organic letters. 22, 4, p. 1585-1588 4 p.

    Research output: Contribution to journal › Article › Research › peer review

  18. External

    Scalable Synthesis of Functionalized Ferrocenyl Azides and Amines Enabled by Flow Chemistry

    Kleoff, M., Schwan, J., Boeser, L., Hartmayer, B., Christmann, M., Sarkar, B. & Heretsch, P., 7 Feb 2020, In: Organic letters. 22, 3, p. 902-907 6 p.

    Research output: Contribution to journal › Article › Research › peer review

  19. External

    Five-Step Synthesis of Yaequinolones J1 and J2

    Schwan, J., Kleoff, M., Heretsch, P. & Christmann, M., 17 Jan 2020, In: Organic letters. 22, 2, p. 675-678 4 p.

    Research output: Contribution to journal › Article › Research › peer review

  20. External

    Synthesis of Swinhoeisterol A, Dankasterone A and B, and Periconiastone A by Radical Framework Reconstruction

    Duecker, F. L., Heinze, R. C. & Heretsch, P., 8 Jan 2020, In: Journal of the American Chemical Society. 142, 1, p. 104-108 5 p.

    Research output: Contribution to journal › Article › Research › peer review

  21. 2019

  22. External

    Contemporary Synthetic Strategies towards Secosteroids, abeo -Steroids, and Related Triterpenes

    Noack, F., Heinze, R. C. & Heretsch, P., May 2019, In: SYNTHESIS-STUTTGART. 51, 10, p. 2039-2057 19 p.

    Research output: Contribution to journal › Article › Research

  23. External

    Rearranged ergostane-type natural products: chemistry, biology, and medicinal aspects

    Duecker, F. L., Reuss, F. & Heretsch, P., 21 Feb 2019, In: Organic and Biomolecular Chemistry. 17, 7, p. 1624-1633 10 p.

    Research output: Contribution to journal › Article › Research

  24. External

    Translation of a Polar Biogenesis Proposal into a Radical Synthetic Approach: Synthesis of Pleurocin A/Matsutakone and Pleurocin B

    Heinze, R. C. & Heretsch, P., 23 Jan 2019, In: Journal of the American Chemical Society. 141, 3, p. 1222-1226 5 p.

    Research output: Contribution to journal › Article › Research › peer review

  25. 2018

  26. External

    Synthesis of Quinolinone Alkaloids via Aryne Insertions into Unsymmetric Imides in Flow

    Schwan, J., Kleoff, M., Hartmayer, B., Heretsch, P. & Christmann, M., 7 Dec 2018, In: Organic Letters. 20, 23, p. 7661-7664 4 p.

    Research output: Contribution to journal › Article › Research › peer review

  27. External

    Photochemical degradation of trypan blue

    Brockman, T., Blanchard, V., Heretsch, P., Brockmann, C. & Bertelmann, E., 10 Apr 2018, In: PLOS ONE. 13, 4, e0195849.

    Research output: Contribution to journal › Article › Research › peer review

  28. External

    Access to 5(6 -> 7)abeo-Steroids through Benzilic Acid Rearrangement of i-Steroids

    Noack, F., Hartmayer, B. & Heretsch, P., 18 Jan 2018, In: Synthesis. 50, 04, p. 809-820 12 p.

    Research output: Contribution to journal › Article › Research › peer review

  29. 2017

  30. Published

    Form Follows Function: Designer Chemistry at the 52nd Bürgenstock Conference

    Heretsch, P., 24 Jul 2017, In: Angewandte Chemie - International Edition. 56, 31, p. 8933-8936 4 p.

    Research output: Contribution to journal › Review article › Research › peer review

  31. Published

    Synthesis of Secosterols as an Arena for C-H Functionalization and C-C Manipulation Tactics

    Heinze, R. C. & Heretsch, P., Jun 2017, In: SYNLETT. 28, 10, p. 1127-1133 7 p.

    Research output: Contribution to journal › Article › Research › peer review

  32. 2016

  33. External

    Synthesis of StrophasterolA Guided by a Proposed Biosynthesis and Innate Reactivity

    Heinze, R. C., Lentz, D. & Heretsch, P., 12 Sept 2016, In: Angewandte Chemie - International Edition. 55, 38, p. 11656-11659 4 p.

    Research output: Contribution to journal › Article › Research › peer review

  34. External

    Total Synthesis of Δ 12-Prostaglandin J 3: Evolution of Synthetic Strategies to a Streamlined Process

    Nicolaou, K. C., Pulukuri, K. K., Yu, R., Rigol, S., Heretsch, P., Grove, C. I., Hale, C. R. H. & ElMarrouni, A., 13 Jun 2016, In: Chemistry - A European Journal. 22, 25, p. 8559-8570 12 p.

    Research output: Contribution to journal › Article › Research › peer review

  35. External

    Synthesis and Biological Investigation of Delta(12)-Prostaglandin J3 (Delta(12)-PGJ(3)) Analogues and Related Compounds

    Nicolaou, K. C., Pulukuri, K. K., Rigol, S., Heretsch, P., Yu, R., Grove, C. I., Hale, C. R. H., ElMarrouni, A., Fetz, V., Broenstrup, M., Aujay, M., Sandoval, J. & Gavrilyuk, J., 25 May 2016, In: Journal of the American Chemical Society. 138, 20, p. 6550-6560 11 p.

    Research output: Contribution to journal › Article › Research › peer review

  36. 2015

  37. Published

    Total Synthesis of Trioxacarcin DC-45-A2

    Nicolaou, K. C., Cai, Q., Qin, B., Petersen, M. T., Mikkelsen, R. J. T. & Heretsch, P., 2 Mar 2015, In: Angewandte Chemie - International Edition. 54, 10, p. 3074-3078

    Research output: Contribution to journal › Article › Research › peer review

  38. Published

    The Veratrum and Solanum alkaloids

    Heretsch, P. & Giannis, A., 2015, In: The Alkaloids. Chemistry and biology. 74, p. 201-32 32 p.

    Research output: Contribution to journal › Review article › Research › peer review

  39. 2014

  40. Published

    Synthesis and Biological Evaluation of QRSTUVWXYZA ' Domains of Maitotoxin

    Nicolaou, K. C., Heretsch, P., Nakamura, T., Rudo, A., Murata, M. & Konoki, K., 19 Nov 2014, In: Journal of the American Chemical Society. 136, 46, p. 16444-16451

    Research output: Contribution to journal › Article › Research › peer review

  41. Published

    Total Synthesis of Delta(12)-Prostaglandin J(3), a Highly Potent and Selective Antileukemic Agent

    Nicolaou, K. C., Heretsch, P., ElMarrouni, A., Hale, C. R. H., Pulukuri, K. K., Kudva, A. K., Narayan, V. & Prabhu, K. S., 22 Sept 2014, In: Angewandte Chemie - International Edition. 53, 39, p. 10443-10447

    Research output: Contribution to journal › Article › Research › peer review

  42. Published

    C-H-Functionalization logic guides the synthesis of a carbacyclopamine analog

    Rabe, S., Moschner, J., Bantzi, M., Heretsch, P. & Giannis, A., 9 Jul 2014, In: Beilstein Journal of Organic Chemistry. 10, p. 1564-1568

    Research output: Contribution to journal › Article › Research › peer review

  43. External

    Cyclopamine and Congeners

    Heretsch, P. & Giannis, A., 19 May 2014, Natural Products in Medicinal Chemistry. Wiley-Blackwell, p. 545-564 20 p.

    Research output: Chapter in book/report/conference proceeding › Contribution to book/anthology › Research › peer review

  44. 2013

  45. Published

    Cyclopamine analogs bearing exocyclic methylenes are highly potent and acid-stable inhibitors of hedgehog signaling

    Moschner, J., Chentsova, A., Eilert, N., Rovardi, I., Heretsch, P. & Giannis, A., 31 Oct 2013, In: Beilstein Journal of Organic Chemistry. 9, p. 2328-2335

    Research output: Contribution to journal › Article › Research › peer review

  46. Published

    Synthesis and antioxidant evaluation of (S,S)- and (R,R)-secoisolariciresinol diglucosides (SDGs)

    Mishra, O. P., Simmons, N., Tyagi, S., Pietrofesa, R., Shuvaev, V. V., Valiulin, R. A., Heretsch, P., Nicolaou, K. C. & Christofidou-Solomidou, M., 1 Oct 2013, In: Bioorganic and Medicinal Chemistry Letters. 23, 19, p. 5325-5328

    Research output: Contribution to journal › Article › Research › peer review

  47. Published

    General Synthetic Approach to Functionalized Dihydrooxepines

    Nicolaou, K. C., Yu, R., Shi, L., Cai, Q., Lu, M. & Heretsch, P., 19 Apr 2013, In: Organic letters. 15, 8, p. 1994-1997

    Research output: Contribution to journal › Article › Research › peer review

  48. 2012

  49. Published

    Synthesis and Biological Evaluation of Epidithio-, Epitetrathio-, and bis-(Methylthio)diketopiperazines: Synthetic Methodology, Enantioselective Total Synthesis of Epicoccin G, 8,8 '-epi-ent-Rostratin B, Gliotoxin, Gliotoxin G, Emethallicin E, and Haematocin and Discovery of New Antiviral and Antimalarial Agents

    Nicolaou, K. C., Lu, M., Totokotsopoulos, S., Heretsch, P., Giguere, D., Sun, Y., Sarlah, D., Nguyen, T. H., Wolf, I. C., Smee, D. F., Day, C. W., Bopp, S. & Winzeler, E. A., 17 Oct 2012, In: Journal of the American Chemical Society. 134, 41, p. 17320-17332

    Research output: Contribution to journal › Article › Research › peer review

  50. Published

    Microbiologically produced carboxylic acids used as building blocks in organic synthesis

    Aurich, A., Specht, R., Müller, R. A., Stottmeister, U., Yovkova, V., Otto, C., Holz, M., Barth, G., Heretsch, P., Thomas, F. A., Sicker, D. & Giannis, A., 2012, In: Subcellular Biochemistry. 64, p. 391-423 33 p.

    Research output: Contribution to journal › Review article › Research › peer review

  51. 2011

  52. Published

    Enantioselective Dichlorination of Allylic Alcohols

    Nicolaou, K. C., Simmons, N. L., Ying, Y., Heretsch, P. M. & Chen, J. S., 1 Jun 2011, In: Journal of the American Chemical Society. 133, 21, p. 8134-8137

    Research output: Contribution to journal › Article › Research › peer review

  53. Published

    Exo-Cyclopamine-a stable and potent inhibitor of hedgehog-signaling

    Heretsch, P., Buettner, A., Tzagkaroulaki, L., Zahn, S., Kirchner, B. & Giannis, A., 2011, In: Chemical communications. 47, 26, p. 7362-7364

    Research output: Contribution to journal › Article › Research › peer review

  54. 2010

  55. Published

    Modulators of the hedgehog signaling pathway

    Heretsch, P., Tzagkaroulaki, L. & Giannis, A., 15 Sept 2010, In: Bioorganic and Medicinal Chemistry. 18, 18, p. 6613-6624

    Research output: Contribution to journal › Review article › Research › peer review

  56. Published

    A Biomimetic Approach to C-nor-D-homo-Steroids

    Heretsch, P., Rabe, S. & Giannis, A., 28 Jul 2010, In: Journal of the American Chemical Society. 132, 29, p. 9968-9969

    Research output: Contribution to journal › Article › Research › peer review

  57. Published

    Cyclopamine and Hedgehog Signaling: Chemistry, Biology, Medical Perspectives

    Heretsch, P., Tzagkaroulaki, L. & Giannis, A., 2010, In: Angewandte Chemie - International Edition. 49, 20, p. 3418-3427

    Research output: Contribution to journal › Review article › Research › peer review

  58. 2009

  59. Published

    Synthesis of All Diastereomers of the Piperidine-Alkaloid Substructure of Cyclopamine

    Heretsch, P., Rabe, S. & Giannis, A., 3 Dec 2009, In: Organic letters. 11, 23, p. 5410-5412

    Research output: Contribution to journal › Article › Research › peer review

  60. Published

    Synthesis of Cyclopamine Using a Biomimetic and Diastereoselective Approach

    Giannis, A., Heretsch, P., Sarli, V. & Stossel, A., 2009, In: Angewandte Chemie - International Edition. 48, 42, p. 7911-7914

    Research output: Contribution to journal › Article › Research › peer review

  61. 2008

  62. Published

    Syntheses with a chiral building block from the citric acid cycle: (2R,3S)-Isocitric acid by fermentation of sunflower oil

    Heretsch, P., Thomas, F., Aurich, A., Krautscheid, H., Sicker, D. & Giannis, A., 2008, In: Angewandte Chemie - International Edition. 47, 10, p. 1958-1960

    Research output: Contribution to journal › Article › Research › peer review

  63. 2007

  64. Published

    An efficient entry to amino-substituted resorcylic acid derivatives for the synthesis of platensimycin and analogues

    Heretsch, P. & Giannis, A., 3 Sept 2007, In: SYNTHESIS-STUTTGART. 17, p. 2614-2616

    Research output: Contribution to journal › Article › Research › peer review