Synthesis of unsaturated lactone moieties by asymmetric hetero Diels-Alder reactions with binaphthol-titanium complexes

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Original languageEnglish
Pages (from-to)1263-1265
Number of pages3
JournalTetrahedron letters
Volume42
Issue number7
Publication statusPublished - 12 Feb 2001

Abstract

Natural products like ratjadone and callystatin A contain an α,β-unsaturated lactone moiety which adds to the biological activity of these compounds. Here we report a rapid and practical access to lactone precursor 3 by an asymmetric hetero Diels-Alder reaction as the key step and its subsequent transformation into a suitable building block 4.

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Synthesis of unsaturated lactone moieties by asymmetric hetero Diels-Alder reactions with binaphthol-titanium complexes. / Quitschalle, Monika; Christmann, Mathias; Bhatt, Ulhas et al.
In: Tetrahedron letters, Vol. 42, No. 7, 12.02.2001, p. 1263-1265.

Research output: Contribution to journalArticleResearchpeer review

Quitschalle M, Christmann M, Bhatt U, Kalesse M. Synthesis of unsaturated lactone moieties by asymmetric hetero Diels-Alder reactions with binaphthol-titanium complexes. Tetrahedron letters. 2001 Feb 12;42(7):1263-1265. doi: 10.1016/S0040-4039(00)02213-9
Quitschalle, Monika ; Christmann, Mathias ; Bhatt, Ulhas et al. / Synthesis of unsaturated lactone moieties by asymmetric hetero Diels-Alder reactions with binaphthol-titanium complexes. In: Tetrahedron letters. 2001 ; Vol. 42, No. 7. pp. 1263-1265.
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